Topic: Male
Journal: Journal of Medicinal Chemistry
Documents
A list of abstracts that contain a topic of "Male" and a journal name of "Journal of Medicinal Chemistry".
Identification and Optimization of Anthranilic Sulfonamides As Novel, Selective Cholecystokinin-2 Receptor Antagonists.
PMID: 17034143
Synthesis and Biological Evaluation of [18f]bicalutamide, 4-[76br]bromobicalutamide, and 4-[76br]bromo-thiobicalutamide As Non-steroidal Androgens for Prostate Cancer Imaging.
PMID: 17328524
Evaluation of Carbon-11-labeled 2beta-carbomethoxy-3beta-[4'-((Z)-2-iodoethenyl)phenyl]nortropane As a Potential Radioligand for Imaging the Serotonin Transporter by Pet.
PMID: 16451060
Novel Tricyclic Compounds Having Acetylene Groups at C-8a and Cyano Enones in Rings A and C: Highly Potent Anti-inflammatory and Cytoprotective Agents.
PMID: 17367124
3d-qsar Studies on Cannabinoid Cb1 Receptor Agonists: G-protein Activation As Biological Data.
PMID: 16420041
Design of Potent, Orally Available Antagonists of the Transient Receptor Potential Vanilloid 1. Structure-activity Relationships of 2-piperazin-1-yl-1h-benzimidazoles.
PMID: 16759115
Synthesis and Biological Evaluation of Chiral Alpha-aminoanilides with Central Antinociceptive Activity.
PMID: 17373780
Evaluation of Basic Amphipathic Peptides for Cellular Delivery of Antisense Peptide Nucleic Acids.
PMID: 16610796
Iron Binding Dendrimers: a Novel Approach for the Treatment of Haemochromatosis.
PMID: 16821777
Neuropeptide Y (Npy) Y4 Receptor Selective Agonists Based on Npy(32-36): Development of an Anorectic Y4 Receptor Selective Agonist with Picomolar Affinity.
PMID: 16610810
Discovery of Aminoquinazolines As Potent, Orally Bioavailable Inhibitors of Lck: Synthesis, Sar, and in Vivo Anti-inflammatory Activity.
PMID: 16970394
1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles: Identification of a Potent Aurora Kinase Inhibitor with a Favorable Antitumor Kinase Inhibition Profile.
PMID: 17125279
Comparison of the Binding of 3-fluoromethyl-7-sulfonyl-1,2,3,4-tetrahydroisoquinolines with Their Isosteric Sulfonamides to the Active Site of Phenylethanolamine N-methyltransferase.
PMID: 16942016
Synthesis and Antifungal Activity of a Novel Series of Alkyldimethylamine Cyanoboranes and Their Derivatives.
PMID: 16884300
Analogues with Fluorescent Leaving Groups for Screening and Selection of Enzymes That Efficiently Hydrolyze Organophosphorus Nerve Agents.
PMID: 16392809
2-[(4-phenylpiperazin-1-yl)methyl]imidazo(Di)azines As Selective D4-ligands. Induction of Penile Erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (Pip3ea), a Potent and Selective D4 Partial Agonist.
PMID: 16789750
Design and Synthesis of Novel Hydrazide-linked Bifunctional Peptides As Delta/Mu Opioid Receptor Agonists and Cck-1/Cck-2 Receptor Antagonists.
PMID: 16509592
Synthesis and Characterization of Potent and Selective Mu-opioid Receptor Antagonists, [Dmt(1), D-2-nal(4)]endomorphin-1 (Antanal-1) and [Dmt(1), D-2-nal(4)]endomorphin-2 (Antanal-2).
PMID: 17266203